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Crystal structure of JAK2 JH1 with type II inhibitor YLIU-04-105-1

Akinori Yoda, Amanda Ceas, Brian Lawney, Catharine Leahy, David M. Weinstock, Dikshat G. Gupta, Haley Cirka, Hwan Geun Choi, Jingyun Dong, Kristen E. Stevenson, Kristen L. Jones, Lei Yang, Loretta S. Li, Matthew L. Arwood, Mingfeng Hao, Nathanael S. Gray, Olivia D. Plana, Shannon K. Harkins, Stevan R. Hubbard, Tinghu Zhang, Yaning Wang, Yao Liu, Zhixiang He, Anniina T. Virtanen, Olli Silvennoinen2023

Crystal structure of JAK2 JH2-V617F in complex with Z902-A1

Jianping Liu, Natalia Nekhotiaeva, Parthasarathy Sampathkumar, Sanna Liukkonen, Stevan R. Hubbard, Anniina T. Virtanen, Maaria Palmroth, Olli Silvennoinen, Teemu Haikarainen2023

Crystal structure of JAK2 JH2-V617F in complex with Reversine

Jianping Liu, Natalia Nekhotiaeva, Parthasarathy Sampathkumar, Sanna Liukkonen, Stevan R. Hubbard, Anniina T. Virtanen, Maaria Palmroth, Olli Silvennoinen, Teemu Haikarainen2023

Crystal structure of JAK2 JH2-V617F in complex with Cdk2 inhibitor IV

Jianping Liu, Natalia Nekhotiaeva, Parthasarathy Sampathkumar, Sanna Liukkonen, Stevan R. Hubbard, Anniina T. Virtanen, Maaria Palmroth, Olli Silvennoinen, Teemu Haikarainen2023

Crystal structure of JAK2 JH2-V617F in complex with Bemcentinib

Jianping Liu, Natalia Nekhotiaeva, Parthasarathy Sampathkumar, Sanna Liukkonen, Stevan R. Hubbard, Anniina T. Virtanen, Maaria Palmroth, Olli Silvennoinen, Teemu Haikarainen2023

Crystal structure of JAK2 JH2-V617F in complex with CB76

Jianping Liu, Natalia Nekhotiaeva, Parthasarathy Sampathkumar, Sanna Liukkonen, Stevan R. Hubbard, Anniina T. Virtanen, Maaria Palmroth, Olli Silvennoinen, Teemu Haikarainen2023

Crystal structure of JAK2 JH2-V617F in complex with HTS-A3

Jianping Liu, Natalia Nekhotiaeva, Parthasarathy Sampathkumar, Sanna Liukkonen, Stevan R. Hubbard, Anniina T. Virtanen, Maaria Palmroth, Olli Silvennoinen, Teemu Haikarainen2023

Crystal structure of JAK2 JH2 in complex with Bemcentinib

Jianping Liu, Parthasarathy Sampathkumar, Sanna Liukkonen, Anniina T. Virtanen, Maaria Palmroth, Olli Silvennoinen, Teemu Haikarainen2023

Crystal structure of JAK2 JH2-V617F in complex with Z902-A3

Jianping Liu, Natalia Nekhotiaeva, Parthasarathy Sampathkumar, Sanna Liukkonen, Stevan R. Hubbard, Anniina T. Virtanen, Maaria Palmroth, Olli Silvennoinen, Teemu Haikarainen2023

Crystal structure of JAK2 JH2 (pseudokinase domain) in complex with HTSA3

Natalia Nekhotiaeva, Parthasarathy Sampathkumar, Sanna Liukkonen, Stevan R. Hubbard, Anniina T. Virtanen, Maaria Palmroth, Olli Silvennoinen, Teemu Haikarainen2023