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Publications information icon
Development of an enzyme-coupled activity assay for Janus kinase 2
inhibitor
screening
Peer-reviewed
Open access
DOI
10.1016/j.slasd.2023.05.001
Pölläniemi, Angelika; Virtanen, Anniina; Silvennoinen, Olli; Haikarainen, Teemu
SLAS discovery
2023
Publications information icon
Methods to Evaluate the Effects of HAT/KAT Inhibition on SIAH2-Driven Reactive Oxygen Species Generation in Helicobacter pylori-Infected Gastric Epithelial Cells
Peer-reviewed
DOI
10.1007/978-1-0716-2788-4_21
Dixit, Pragyesh; Kokate, Shrikant Babanrao; Rath, Suvasmita; Das, Lopamudra; Chakraborty, Debashish;...
Methods in Molecular Biology
2023
Publications information icon
Discovery of MINC1, a GTPase-Activating Protein Small Molecule
Inhibitor
, Targeting MgcRacGAP
Peer-reviewed
Open access
van Adrichem, Arjan J.; Fagerholm, Annika; Turunen, Laura; Lehto, Anna; Saarela, Jani; Koskinen, Ari...
Combinatorial chemistry and high throughput screening
2015
Publications information icon
Electrophysiological determination of phosphodiesterase-6
inhibitor
inhibition constants in intact mouse retina
Peer-reviewed
Open access
DOI
10.1016/j.taap.2018.03.002
Turunen, Teemu T.; Koskelainen, Ari
Toxicology and Applied Pharmacology
2018
Publications information icon
PP2A
inhibitor
PME-1 drives kinase inhibitor resistance in glioma cells
Peer-reviewed
DOI
10.1158/0008-5472.can-16-1134
Kaur, Amanpreet; Denisova, Oxana V.; Qiao, Xi; Jumppanen, Mikael; Peuhu, Emilia; Ahmed, Shafiq U.; R...
Cancer research
2016
Publications information icon
EGFR
inhibitor
and chemotherapy combinations for acquired TKI resistance in EGFR-mutant NSCLC models
Peer-reviewed
DOI
10.1007/s12032-015-0627-6
Laurila, Niina; Koivunen, Jussi P.
Medical oncology
2015
Publications information icon
Efficacy of Novel CA IX
Inhibitor
s in Biological Models
Peer-reviewed
DOI
10.1007/978-3-030-12780-0_18
Kazokaite, Justina;Becker, Holger M.;Barker, Harlan R.;Aspatwar, Ashok;Parkkila, Seppo;Dubois, Ludwi...
Springer
2019
Publications information icon
Adverse effects of an aldosterone synthase (CYP11B2)
inhibitor
, fadrozole (FAD286), on inflamed rat colon
Peer-reviewed
Open access
DOI
10.1111/bcpt.13918
Launonen, Hanna; Luiskari, Lotta; Linden, Jere; Siltari, Aino; Salmenkari, Hanne; Korpela, Riitta; V...
Basic and clinical pharmacology and toxicology
2023
Publications information icon
In vivo and in vitro inhibition of osteosarcoma growth by the pan Bcl-2
inhibitor
AT-101
Peer-reviewed
DOI
10.1007/s10637-019-00827-y
Masuelli, Laura; Benvenuto, Monica; Izzi, Valerio; Zago, Erika; Mattera, Rosanna; Cerbelli, Bruna; P...
Investigational new drugs
2019
Publications information icon
Human Mono-ADP-ribosyl transferases :
inhibitor
development for new potential drug targets
Murthy, Sudarshan Narasimha
Faculty of biochemisty and molecular medicine
2020
Development of an enzyme-coupled activity assay for Janus kinase 2
inhibitor
screening
Peer-reviewed
Open access
DOI
10.1016/j.slasd.2023.05.001
2023
Methods to Evaluate the Effects of HAT/KAT Inhibition on SIAH2-Driven Reactive Oxygen Species Generation in Helicobacter pylori-Infected Gastric Epithelial Cells
Peer-reviewed
DOI
10.1007/978-1-0716-2788-4_21
2023
Discovery of MINC1, a GTPase-Activating Protein Small Molecule
Inhibitor
, Targeting MgcRacGAP
Peer-reviewed
Open access
2015
Electrophysiological determination of phosphodiesterase-6
inhibitor
inhibition constants in intact mouse retina
Peer-reviewed
Open access
DOI
10.1016/j.taap.2018.03.002
2018
PP2A
inhibitor
PME-1 drives kinase inhibitor resistance in glioma cells
Peer-reviewed
DOI
10.1158/0008-5472.can-16-1134
2016
EGFR
inhibitor
and chemotherapy combinations for acquired TKI resistance in EGFR-mutant NSCLC models
Peer-reviewed
DOI
10.1007/s12032-015-0627-6
2015
Efficacy of Novel CA IX
Inhibitor
s in Biological Models
Peer-reviewed
DOI
10.1007/978-3-030-12780-0_18
2019
Adverse effects of an aldosterone synthase (CYP11B2)
inhibitor
, fadrozole (FAD286), on inflamed rat colon
Peer-reviewed
Open access
DOI
10.1111/bcpt.13918
2023
In vivo and in vitro inhibition of osteosarcoma growth by the pan Bcl-2
inhibitor
AT-101
Peer-reviewed
DOI
10.1007/s10637-019-00827-y
2019
Human Mono-ADP-ribosyl transferases :
inhibitor
development for new potential drug targets
2020
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