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Pyrazinyl-Substituted Aminoazoles as Covalent Inhibitors of Thrombin: Synthesis, Structure, and Anticoagulant Properties

Year of publication

2024

Authors

Imberg, Lukas; Siutkina, Alena I; Erbacher, Catharina; Schmidt, Judith; Broekmans, Darius F; Ovsepyan, Ruzanna A; Daniliuc, Constantin G; de Oliveira, Ellen Goncalves; Serafim, Mateus Sa Magalhaes; O'Donoghue, Anthony J; Pillaiyar, Thanigaimalai; Panteleev, Mikhail A; Poso, Antti; Kalinina, Svetlana A; Bermudez, Marcel; Nekipelov, Katrin; Bendas, Gerd; Karst, Uwe; Kalinin, Dmitrii V
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Organizations and authors

Publication type

Publication format

Article

Parent publication type

Journal

Article type

Original article

Audience

Scientific

Peer-reviewed

Peer-Reviewed

MINEDU's publication type classification code

A1 Journal article (refereed), original research

Publication channel information

Volume

2025; 8

Issue

1

Pages

146-172

​Publication forum

88746

​Publication forum level

1

Open access

Open access in the publisher’s service

No

Open access of publication channel

Partially open publication channel

Self-archived

No

Other information

Fields of science

Pharmacy

Internationality of the publisher

International

Language

English

International co-publication

Yes

Co-publication with a company

No

DOI

10.1021/acsptsci.4c00515

The publication is included in the Ministry of Education and Culture’s Publication data collection

Yes